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8-Cl-cAMP

8- Chloroadenosine- 3', 5'- cyclic monophosphate ( 8-Cl-cAMP ), sodium salt
Site-selective PKA agonist
Cat. No.: C 007
    
CAS No.: [124705-03-9]
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Product Name Price (net) Qty
Cat. No.: C 007-10
Unit: 10 µmol / ~3.9 mg
$96.00
For metabolites of 8-Cl-cAMP please refer to Cat. No. C 008; for related items or other salt forms please inquire. Site-selective cyclic AMP analogue with high selectivity for protein kinase A type I. Induces growth inhibition and differentiation in cultured cancer cell lines and has been tested in several clinical trials already. Detailed technical information and updated reference available on request. Reference: Schwede et al., Pharmacol. Ther., 87, 199 – 226 (2000).
Cat. No. C 007
CAS number [124705-03-9]
Purity > 99% HPLC
Salt form Sodium
Storage temperature -20°C / -4°F
Molecular formula C₁₀H₁₀ClN₅O₆P · Na
Molecular weight [g/mol] 385,6
Modifications 8-cAMP
Target PKA (cAK) Activator
Lipophilicity 1.31
Absorption max [nm] 262
Molar extinction coefficient ε [L·mol⁻¹·cm⁻¹] 17000
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