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Alternative structural projections:

8-pCPT-2'-O-Me-cAMP

8- (4- Chlorophenylthio)- 2'- O- methyladenosine- 3', 5'- cyclic monophosphate ( 8-pCPT-2'-O-Me-cAMP / 8-CPT-2'-O-Me-cAMP / 8-CPT-2Me-cAMP / "007" ), sodium salt
Specific, membrane-permeant Epac activator
Cat. No.: C 041
    
CAS No.: [634207-53-7]
Shipping: ambient
Product Name Price (net) Qty
Cat. No.: C 041-05
Unit: 5 µmol / ~2.5 mg
$235.00

For other salt forms please inquire. Specific activator of the exchange protein activated by cyclic AMP (Epac) or cAMP-GEF, respectively, which does not activate protein kinase A. High lipophilicity and membrane permeability, as well as increased PDE stability. Potential metabolites are offered as well. Detailed technical information and updated references available. References: Enserink et al., Nature Cell Biol., 4, 901 - 906 (2002); Kang et al., J. Biol. Chem., 278, 8279 - 8285 (2003); Christensen et al., J. Biol. Chem., 278, 35394 - 35402 (2003).

Cat. No. C 041
CAS number [634207-53-7]
Purity >98% HPLC
Salt form Sodium
Storage temperature -20°C / -4°F
Molecular formula C₁₇H₁₆ClN₅O₆PS · Na
Molecular weight [g/mol] 507.8
Modifications 8-cAMP, 2'-cAMP
Target Epac Activator
Lipophilicity 2.95
Absorption max [nm] 282
Molar extinction coefficient ε [L·mol⁻¹·cm⁻¹] 16000
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