For other salt forms please inquire. Specific activator of the exchange protein activated by cyclic AMP (Epac) or cAMP-GEF, respectively, which does not activate protein kinase A. High lipophilicity and membrane permeability, as well as increased PDE stability. Potential metabolites are offered as well. Detailed technical information and updated references available. References: Enserink et al., Nature Cell Biol., 4, 901 - 906 (2002); Kang et al., J. Biol. Chem., 278, 8279 - 8285 (2003); Christensen et al., J. Biol. Chem., 278, 35394 - 35402 (2003).
Cat. No. | C 041 |
CAS number | [634207-53-7] |
Purity | >98% HPLC |
Salt form | Sodium |
Storage temperature | -20°C / -4°F |
Molecular formula | C₁₇H₁₆ClN₅O₆PS · Na |
Molecular weight [g/mol] | 507.8 |
Modifications | 8-cAMP, 2'-cAMP |
Target | Epac Activator |
Lipophilicity | 2.95 |
Absorption max [nm] | 282 |
Molar extinction coefficient ε [L·mol⁻¹·cm⁻¹] | 16000 |