C₁₇H₁₆ClN₅O₆PS^.Na; MW 507.8; λ_max 282 nm; ε 16000; sodium salt; purity > 98% HPLC. For other salt forms please inquire. Specific activator of the exchange protein activated by cyclic AMP (Epac) or cAMP-GEF, respectively, which does not activate protein kinase A. High lipophilicity and membrane permeability, as well as increased PDE stability. Potential metabolites are offered as well. Detailed technical information and updated references available. References: Enserink et al., Nature Cell Biol., 4, 901 - 906 (2002); Kang et al., J. Biol. Chem., 278, 8279 - 8285 (2003); Christensen et al., J. Biol. Chem., 278, 35394 - 35402 (2003).

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