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ESI-09

3- [5- (tert.-Butyl)isoxazol- 3- yl]- 2- [2- (3- chlorophenyl)hydrazono]- 3- oxopropanenitrile ( ESI-09 )
Membrane-permeant inhibitor of Epac 1 and Epac 2
Cat. No.: B 133
    
CAS No.: [263707-16-0]
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Product Name Price (net) Qty
Cat. No.: B 133-05
Unit: 5 µmol / ~1.7 mg
$345.00
According to Almahariq et al. (2013) ESI-09 is a membrane-permeant inhibitor of Epac 1 and Epac 2. Detailed technical information available. Reference: Almahariq et al., Mol. Pharmacol., 83, 122 - 128 (2013).
Cat. No. B 133
CAS number [263707-16-0]
Purity > 95% HPLC
Storage temperature -20°C / -4°F
Molecular formula C₁₆H₁₅ClN₄O₂
Molecular weight [g/mol] 330,8
Target Epac Inhibitor
Absorption max [nm] 384
Molar extinction coefficient ε [L·mol⁻¹·cm⁻¹] 25300
  • 1. Almahariq M., Tsalkova T., Mei F. C., Chen H., Zhou J., Sastry S. K., Schwede F.Cheng X., Mol. Pharmacol., 83, 122 - 128 (2013), "A Novel EPAC Specific Inhibitor Suppresses Pancreatic Cancer Cell Migration and Invasion"
  • 2. Rehmann H., Sci. Rep., 3: 3032, 0, 0 - 0 (2013), "Epac-Inhibitors: Facts and Artefacts"